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Journal Abstract Search


132 related items for PubMed ID: 28409931

  • 1. 1-(4-[18F]Fluorobenzyl)-4-[(tetrahydrofuran-2-yl)methyl]piperazine: A Novel Suitable Radioligand with Low Lipophilicity for Imaging σ1 Receptors in the Brain.
    He Y, Xie F, Ye J, Deuther-Conrad W, Cui B, Wang L, Lu J, Steinbach J, Brust P, Huang Y, Lu J, Jia H.
    J Med Chem; 2017 May 25; 60(10):4161-4172. PubMed ID: 28409931
    [Abstract] [Full Text] [Related]

  • 2. Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising σ1 receptor imaging agent.
    Chen YY, Wang X, Zhang JM, Deuther-Conrad W, Zhang XJ, Huang Y, Li Y, Ye JJ, Cui MC, Steinbach J, Brust P, Liu BL, Jia HM.
    Bioorg Med Chem; 2014 Oct 01; 22(19):5270-8. PubMed ID: 25189691
    [Abstract] [Full Text] [Related]

  • 3. 18 F-Labeled benzylpiperazine derivatives as highly selective ligands for imaging σ1 receptor with positron emission tomography.
    Ye J, Wang L, Deuther-Conrad W, Chen Y, Zhang X, Zhang J, Huang Y, Brust P, Jia H.
    J Labelled Comp Radiopharm; 2019 Jun 30; 62(8):425-437. PubMed ID: 30991462
    [Abstract] [Full Text] [Related]

  • 4. Synthesis and evaluation of new 1-oxa-8-azaspiro[4.5]decane derivatives as candidate radioligands for sigma-1 receptors.
    Tian J, He Y, Deuther-Conrad W, Fu H, Xie F, Zhang Y, Wang T, Zhang X, Zhang J, Brust P, Huang Y, Jia H.
    Bioorg Med Chem; 2020 Jul 15; 28(14):115560. PubMed ID: 32616183
    [Abstract] [Full Text] [Related]

  • 5. Synthesis and evaluation of fluorine-18-labeled SA4503 as a selective sigma1 receptor ligand for positron emission tomography.
    Kawamura K, Tsukada H, Shiba K, Tsuji C, Harada N, Kimura Y, Ishiwata K.
    Nucl Med Biol; 2007 Jul 15; 34(5):571-7. PubMed ID: 17591557
    [Abstract] [Full Text] [Related]

  • 6. Synthesis and in vivo evaluation of [18F]N-(2-benzofuranylmethyl)-N'-[4-(2-fluoroethoxy)benzyl]piperazine, a novel σ1 receptor PET imaging agent.
    Moussa IA, Banister SD, Giboureau N, Meikle SR, Kassiou M.
    Bioorg Med Chem Lett; 2011 Nov 15; 21(22):6820-3. PubMed ID: 21962578
    [Abstract] [Full Text] [Related]

  • 7. Synthesis and evaluation of novel (18)F-labeled spirocyclic piperidine derivatives as σ1 receptor ligands for positron emission tomography imaging.
    Li Y, Wang X, Zhang J, Deuther-Conrad W, Xie F, Zhang X, Liu J, Qiao J, Cui M, Steinbach J, Brust P, Liu B, Jia H.
    J Med Chem; 2013 May 09; 56(9):3478-91. PubMed ID: 23566245
    [Abstract] [Full Text] [Related]

  • 8. Synthesis and evaluation of a (18) F-labeled 4-phenylpiperidine-4-carbonitrile radioligand for σ1 receptor imaging.
    Ye J, Wang X, Deuther-Conrad W, Zhang J, Li J, Zhang X, Wang L, Steinbach J, Brust P, Jia H.
    J Labelled Comp Radiopharm; 2016 Jul 09; 59(9):332-9. PubMed ID: 27277387
    [Abstract] [Full Text] [Related]

  • 9. Synthesis and biological evaluation of ¹⁸F labeled fluoro-oligo-ethoxylated 4-benzylpiperazine derivatives for sigma-1 receptor imaging.
    Wang X, Li Y, Deuther-Conrad W, Xie F, Chen X, Cui MC, Zhang XJ, Zhang JM, Steinbach J, Brust P, Liu BL, Jia HM.
    Bioorg Med Chem; 2013 Jan 01; 21(1):215-22. PubMed ID: 23199475
    [Abstract] [Full Text] [Related]

  • 10. (18)F-Labeled 1,4-Dioxa-8-azaspiro[4.5]decane Derivative: Synthesis and Biological Evaluation of a σ1 Receptor Radioligand with Low Lipophilicity as Potent Tumor Imaging Agent.
    Xie F, Bergmann R, Kniess T, Deuther-Conrad W, Mamat C, Neuber C, Liu B, Steinbach J, Brust P, Pietzsch J, Jia H.
    J Med Chem; 2015 Jul 23; 58(14):5395-407. PubMed ID: 26090686
    [Abstract] [Full Text] [Related]

  • 11. Synthesis and evaluation of [18F]fluoroethyl SA4503 as a PET ligand for the sigma receptor.
    Elsinga PH, Kawamura K, Kobayashi T, Tsukada H, Senda M, Vaalburg W, Ishiwata K.
    Synapse; 2002 Mar 15; 43(4):259-67. PubMed ID: 11835521
    [Abstract] [Full Text] [Related]

  • 12. Chiral resolution of serial potent and selective σ1 ligands and biological evaluation of (-)-[18F]TZ3108 in rodent and the nonhuman primate brain.
    Yue X, Jin H, Luo Z, Liu H, Zhang X, McSpadden ED, Tian L, Flores HP, Perlmutter JS, Parsons SM, Tu Z.
    Bioorg Med Chem; 2017 Feb 15; 25(4):1533-1542. PubMed ID: 28129990
    [Abstract] [Full Text] [Related]

  • 13. Novel cyclopentadienyl tricarbonyl (99m)tc complexes containing 1-piperonylpiperazine moiety: potential imaging probes for sigma-1 receptors.
    Wang X, Li D, Deuther-Conrad W, Lu J, Xie Y, Jia B, Cui M, Steinbach J, Brust P, Liu B, Jia H.
    J Med Chem; 2014 Aug 28; 57(16):7113-25. PubMed ID: 25073047
    [Abstract] [Full Text] [Related]

  • 14. Design, synthesis, and structure-affinity relationships of regioisomeric N-benzyl alkyl ether piperazine derivatives as sigma-1 receptor ligands.
    Moussa IA, Banister SD, Beinat C, Giboureau N, Reynolds AJ, Kassiou M.
    J Med Chem; 2010 Aug 26; 53(16):6228-39. PubMed ID: 20662542
    [Abstract] [Full Text] [Related]

  • 15. Sigma1 and sigma2 receptor binding affinity and selectivity of SA4503 and fluoroethyl SA4503.
    Lever JR, Gustafson JL, Xu R, Allmon RL, Lever SZ.
    Synapse; 2006 May 26; 59(6):350-8. PubMed ID: 16463398
    [Abstract] [Full Text] [Related]

  • 16. Evaluation of 18F-labeled benzodioxine piperazine-based dopamine D4 receptor ligands: lipophilicity as a determinate of nonspecific binding.
    Kügler F, Sihver W, Ermert J, Hübner H, Gmeiner P, Prante O, Coenen HH.
    J Med Chem; 2011 Dec 22; 54(24):8343-52. PubMed ID: 22039961
    [Abstract] [Full Text] [Related]

  • 17. Positron Emission Tomography Imaging Evaluation of a Novel 18F-Labeled Sigma-1 Receptor Radioligand in Cynomolgus Monkeys.
    Jia H, Cai Z, Holden D, He Y, Lin SF, Li S, Baum E, Shirali A, Kapinos M, Gao H, Ropchan J, Huang Y.
    ACS Chem Neurosci; 2020 Jun 03; 11(11):1673-1681. PubMed ID: 32356969
    [Abstract] [Full Text] [Related]

  • 18. Comparison of 4 radiolabeled antagonists for serotonin 5-HT(7) receptor neuroimaging: toward the first PET radiotracer.
    Lemoine L, Andries J, Le Bars D, Billard T, Zimmer L.
    J Nucl Med; 2011 Nov 03; 52(11):1811-8. PubMed ID: 21990574
    [Abstract] [Full Text] [Related]

  • 19. Evaluation of (+)-p-[11C]methylvesamicol for mapping sigma1 receptors: a comparison with [11C]SA4503.
    Ishiwata K, Kawamura K, Yajima K, QingGeLeTu, Mori H, Shiba K.
    Nucl Med Biol; 2006 May 03; 33(4):543-8. PubMed ID: 16720247
    [Abstract] [Full Text] [Related]

  • 20. Design and Investigation of a [18F]-Labeled Benzamide Derivative as a High Affinity Dual Sigma Receptor Subtype Radioligand for Prostate Tumor Imaging.
    Yang D, Comeau A, Bowen WD, Mach RH, Ross BD, Hong H, Van Dort ME.
    Mol Pharm; 2017 Mar 06; 14(3):770-780. PubMed ID: 28135101
    [Abstract] [Full Text] [Related]


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