These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


Pubmed for Handhelds

PUBMED FOR HANDHELDS

Journal Abstract Search

163 related items for PubMed ID: 29784274

  • 1. Chiral analogues of (+)-cyclazosin as potent α1B-adrenoceptor selective antagonist.
    Sagratini G, Buccioni M, Marucci G, Poggesi E, Skorski M, Costanzi S, Giardinà D.
    Bioorg Med Chem; 2018 Jul 23; 26(12):3502-3513. PubMed ID: 29784274
    [Abstract] [Full Text] [Related]

  • 2. Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.
    Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D.
    Bioorg Med Chem; 2007 Mar 15; 15(6):2334-45. PubMed ID: 17276073
    [Abstract] [Full Text] [Related]

  • 3. Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist.
    Giardinà D, Crucianelli M, Romanelli R, Leonardi A, Poggesi E, Melchiorre C.
    J Med Chem; 1996 Nov 08; 39(23):4602-7. PubMed ID: 8917649
    [Abstract] [Full Text] [Related]

  • 4. (+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues.
    Marucci G, Angeli P, Buccioni M, Gulini U, Melchiorre C, Sagratini G, Testa R, Giardinà D.
    Eur J Pharmacol; 2005 Oct 17; 522(1-3):100-7. PubMed ID: 16213480
    [Abstract] [Full Text] [Related]

  • 5. Synthesis and α1-adrenoceptor antagonist activity of tamsulosin analogues.
    Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Poggesi E, Giardinà D.
    Eur J Med Chem; 2010 Dec 17; 45(12):5800-7. PubMed ID: 20934789
    [Abstract] [Full Text] [Related]

  • 6. Simultaneous activation of the α1A-, α1B- and α1D-adrenoceptor subtypes in the nucleus accumbens reduces accumbal dopamine efflux in freely moving rats.
    Aono Y, Taguchi H, Saigusa T, Uchida T, Takada K, Takiguchi H, Shirakawa T, Shimizu N, Koshikawa N, Cools AR.
    Behav Pharmacol; 2015 Feb 17; 26(1-2):73-80. PubMed ID: 25438092
    [Abstract] [Full Text] [Related]

  • 7.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 8.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 9. Searching for cyclazosin analogues as alpha(1B)-adrenoceptor antagonists.
    Giardinà D, Polimanti O, Sagratini G, Angeli P, Gulini U, Marucci G, Melchiorre C, Poggesi E, Leonardi A.
    Farmaco; 2003 Jul 17; 58(7):477-87. PubMed ID: 12818686
    [Abstract] [Full Text] [Related]

  • 10. The affinity and selectivity of α-adrenoceptor antagonists, antidepressants, and antipsychotics for the human α1A, α1B, and α1D-adrenoceptors.
    Proudman RGW, Pupo AS, Baker JG.
    Pharmacol Res Perspect; 2020 Aug 17; 8(4):e00602. PubMed ID: 32608144
    [Abstract] [Full Text] [Related]

  • 11.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 12.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 13. Receptor binding profile of cyclazosin, a new alpha 1B-adrenoceptor antagonist.
    Giardinà D, Crucianelli M, Melchiorre C, Taddei C, Testa R.
    Eur J Pharmacol; 1995 Dec 04; 287(1):13-6. PubMed ID: 8666020
    [Abstract] [Full Text] [Related]

  • 14. Indolylpiperidine derivatives as potent and selective α1B adrenoceptor antagonists.
    Hayashi R, Ohmori E, Moriwaki M, Kumagai H, Isogaya M.
    Bioorg Med Chem Lett; 2015 Sep 15; 25(18):3921-3. PubMed ID: 26238322
    [Abstract] [Full Text] [Related]

  • 15.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 16.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 17. 1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: structure-affinity/activity relationship at alpha1-adrenoceptor subtypes and at 5-HT1A receptors.
    Franchini S, Prandi A, Baraldi A, Sorbi C, Tait A, Buccioni M, Marucci G, Cilia A, Pirona L, Fossa P, Cichero E, Brasili L.
    Eur J Med Chem; 2010 Sep 15; 45(9):3740-51. PubMed ID: 20605276
    [Abstract] [Full Text] [Related]

  • 18. Differential antagonism by conotoxin rho-TIA of contractions mediated by distinct alpha1-adrenoceptor subtypes in rat vas deferens, spleen and aorta.
    Lima V, Mueller A, Kamikihara SY, Raymundi V, Alewood D, Lewis RJ, Chen Z, Minneman KP, Pupo AS.
    Eur J Pharmacol; 2005 Jan 31; 508(1-3):183-92. PubMed ID: 15680270
    [Abstract] [Full Text] [Related]

  • 19. Absolute configuration of the alpha (1B)-adrenoceptor antagonist (+)-cyclazosin.
    Giardinà D, Sagratini G, Grelli M, Gulini U, Melchiorre C, Antolini L.
    Farmaco; 2004 Dec 31; 59(12):965-9. PubMed ID: 15598431
    [Abstract] [Full Text] [Related]

  • 20. Affinity of serotonin receptor antagonists and agonists to recombinant and native alpha1-adrenoceptor subtypes.
    Yoshio R, Taniguchi T, Itoh H, Muramatsu I.
    Jpn J Pharmacol; 2001 Jun 31; 86(2):189-95. PubMed ID: 11459121
    [Abstract] [Full Text] [Related]

    Page: [Next] [New Search]
    of 9.