These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


Pubmed for Handhelds

PUBMED FOR HANDHELDS

Journal Abstract Search

323 related items for PubMed ID: 29880250

  • 1. Identification of novel thiazolo[5,4-d]pyrimidine derivatives as human A1 and A2A adenosine receptor antagonists/inverse agonists.
    Varano F, Catarzi D, Falsini M, Vincenzi F, Pasquini S, Varani K, Colotta V.
    Bioorg Med Chem; 2018 Jul 23; 26(12):3688-3695. PubMed ID: 29880250
    [Abstract] [Full Text] [Related]

  • 2.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 3. 7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: structural investigations at the 5-position to target human A₁ and A(2A) adenosine receptors. Molecular modeling and pharmacological studies.
    Squarcialupi L, Colotta V, Catarzi D, Varano F, Betti M, Varani K, Vincenzi F, Borea PA, Porta N, Ciancetta A, Moro S.
    Eur J Med Chem; 2014 Sep 12; 84():614-27. PubMed ID: 25063944
    [Abstract] [Full Text] [Related]

  • 4.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 5. 5-Substituted 2-benzylidene-1-tetralone analogues as A1 and/or A2A antagonists for the potential treatment of neurological conditions.
    Janse van Rensburg HD, Terre'Blanche G, van der Walt MM, Legoabe LJ.
    Bioorg Chem; 2017 Oct 12; 74():251-259. PubMed ID: 28881253
    [Abstract] [Full Text] [Related]

  • 6. Targeting adenosine receptors with coumarins: synthesis and binding activities of amide and carbamate derivatives.
    Matos MJ, Gaspar A, Kachler S, Klotz KN, Borges F, Santana L, Uriarte E.
    J Pharm Pharmacol; 2013 Jan 12; 65(1):30-4. PubMed ID: 23215685
    [Abstract] [Full Text] [Related]

  • 7.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 8. Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations at the 2-, 5- and 7-positions to enhance affinity and tune selectivity.
    Varano F, Catarzi D, Falsini M, Dal Ben D, Buccioni M, Marucci G, Volpini R, Colotta V.
    Bioorg Med Chem Lett; 2019 Feb 15; 29(4):563-569. PubMed ID: 30638876
    [Abstract] [Full Text] [Related]

  • 9.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 10. Carbamate substituted 2-amino-4,6-diphenylpyrimidines as adenosine receptor antagonists.
    Robinson SJ, Petzer JP, Rousseau AL, Terre'Blanche G, Petzer A, Lourens ACU.
    Bioorg Med Chem Lett; 2016 Feb 01; 26(3):734-738. PubMed ID: 26776359
    [Abstract] [Full Text] [Related]

  • 11.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 12.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 13.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 14. Overcoming the genotoxicity of a pyrrolidine substituted arylindenopyrimidine as a potent dual adenosine A(2A)/A(1) antagonist by minimizing bioactivation to an iminium ion reactive intermediate.
    Lim HK, Chen J, Sensenhauser C, Cook K, Preston R, Thomas T, Shook B, Jackson PF, Rassnick S, Rhodes K, Gopaul V, Salter R, Silva J, Evans DC.
    Chem Res Toxicol; 2011 Jul 18; 24(7):1012-30. PubMed ID: 21667953
    [Abstract] [Full Text] [Related]

  • 15. Synthesis and evaluation of methoxy substituted 2-benzoyl-1-benzofuran derivatives as lead compounds for the development adenosine A1 and/or A2A receptor antagonists.
    Janse van Rensburg HD, Legoabe LJ, Terre'Blanche G, Aucamp J.
    Bioorg Chem; 2020 Jan 18; 94():103459. PubMed ID: 31818481
    [Abstract] [Full Text] [Related]

  • 16. Novel 8-amino-1,2,4-triazolo[4,3-a]pyrazin-3-one derivatives as potent human adenosine A1 and A2A receptor antagonists. Evaluation of their protective effect against β-amyloid-induced neurotoxicity in SH-SY5Y cells.
    Falsini M, Catarzi D, Varano F, Dal Ben D, Marucci G, Buccioni M, Volpini R, Di Cesare Mannelli L, Ghelardini C, Colotta V.
    Bioorg Chem; 2019 Jun 18; 87():380-394. PubMed ID: 30913470
    [Abstract] [Full Text] [Related]

  • 17. Selectivity is species-dependent: Characterization of standard agonists and antagonists at human, rat, and mouse adenosine receptors.
    Alnouri MW, Jepards S, Casari A, Schiedel AC, Hinz S, Müller CE.
    Purinergic Signal; 2015 Sep 18; 11(3):389-407. PubMed ID: 26126429
    [Abstract] [Full Text] [Related]

  • 18. 2-Aminopyrimidines as dual adenosine A1/A2A antagonists.
    Robinson SJ, Petzer JP, Terre'Blanche G, Petzer A, van der Walt MM, Bergh JJ, Lourens AC.
    Eur J Med Chem; 2015 Nov 02; 104():177-88. PubMed ID: 26462195
    [Abstract] [Full Text] [Related]

  • 19.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

  • 20.
    ; . PubMed ID:
    [No Abstract] [Full Text] [Related]

    Page: [Next] [New Search]
    of 17.