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PUBMED FOR HANDHELDS

Journal Abstract Search


672 related items for PubMed ID: 33078877

  • 1. Synthesis, antimicrobial evaluation, DNA gyrase inhibition, and in silico pharmacokinetic studies of novel quinoline derivatives.
    El-Shershaby MH, El-Gamal KM, Bayoumi AH, El-Adl K, Ahmed HEA, Abulkhair HS.
    Arch Pharm (Weinheim); 2021 Feb; 354(2):e2000277. PubMed ID: 33078877
    [Abstract] [Full Text] [Related]

  • 2. Molecular docking, discovery, synthesis, and pharmacological properties of new 6-substituted-2-(3-phenoxyphenyl)-4-phenyl quinoline derivatives; an approach to developing potent DNA gyrase inhibitors/antibacterial agents.
    Alagumuthu M, Arumugam S.
    Bioorg Med Chem; 2017 Feb 15; 25(4):1448-1455. PubMed ID: 28094220
    [Abstract] [Full Text] [Related]

  • 3. Antimicrobial evaluation of thiadiazino and thiazolo quinoxaline hybrids as potential DNA gyrase inhibitors; design, synthesis, characterization and morphological studies.
    Ammar YA, Farag AA, Ali AM, Hessein SA, Askar AA, Fayed EA, Elsisi DM, Ragab A.
    Bioorg Chem; 2020 Jun 15; 99():103841. PubMed ID: 32325335
    [Abstract] [Full Text] [Related]

  • 4. Novel 1,2,4-oxadiazole-chalcone/oxime hybrids as potential antibacterial DNA gyrase inhibitors: Design, synthesis, ADMET prediction and molecular docking study.
    Ibrahim TS, Almalki AJ, Moustafa AH, Allam RM, Abuo-Rahma GEA, El Subbagh HI, Mohamed MFA.
    Bioorg Chem; 2021 Jun 15; 111():104885. PubMed ID: 33838559
    [Abstract] [Full Text] [Related]

  • 5. Targeted potent antimicrobial benzochromene-based analogues: Synthesis, computational studies, and inhibitory effect against 14α-Demethylase and DNA Gyrase.
    Fouda AM, Hassan AH, Eliwa EM, Ahmed HEA, Al-Dies AM, Omar AM, Nassar HS, Halawa AH, Aljuhani N, El-Agrody AM.
    Bioorg Chem; 2020 Dec 15; 105():104387. PubMed ID: 33130344
    [Abstract] [Full Text] [Related]

  • 6. Design, synthesis, and antibacterial evaluation of new quinoline-1,3,4-oxadiazole and quinoline-1,2,4-triazole hybrids as potential inhibitors of DNA gyrase and topoisomerase IV.
    Hofny HA, Mohamed MFA, Gomaa HAM, Abdel-Aziz SA, Youssif BGM, El-Koussi NA, Aboraia AS.
    Bioorg Chem; 2021 Jul 15; 112():104920. PubMed ID: 33910078
    [Abstract] [Full Text] [Related]

  • 7. One-pot synthesis and molecular docking of some new spiropyranindol-2-one derivatives as immunomodulatory agents and in vitro antimicrobial potential with DNA gyrase inhibitor.
    Salem MA, Ragab A, Askar AA, El-Khalafawy A, Makhlouf AH.
    Eur J Med Chem; 2020 Feb 15; 188():111977. PubMed ID: 31927313
    [Abstract] [Full Text] [Related]

  • 8. Antimicrobial Activity of New 2-Thioxo-benzo[g]quinazolin-4(3H)-one Derivatives.
    Al-Salahi R, Abuelizz HA, Dib RE, Marzouk M, Alshammari MB.
    Med Chem; 2016 Feb 15; 13(1):85-92. PubMed ID: 27306606
    [Abstract] [Full Text] [Related]

  • 9. Construction and Docking Studies of Novel Pyrimido[4,5-b]quinolines as Antimicrobial Agents.
    Bakr RB, El Azab IH, Elkanzi NAA.
    Chem Biodivers; 2024 Jun 15; 21(6):e202400200. PubMed ID: 38570192
    [Abstract] [Full Text] [Related]

  • 10. Synthesis, and antibacterial activity of novel 4,5-dihydro-1H-pyrazole derivatives as DNA gyrase inhibitors.
    Liu JJ, Sun J, Fang YB, Yang YA, Jiao RH, Zhu HL.
    Org Biomol Chem; 2014 Feb 14; 12(6):998-1008. PubMed ID: 24382549
    [Abstract] [Full Text] [Related]

  • 11. Development and radiosterilization of new hydrazono-quinoline hybrids as DNA gyrase and topoisomerase IV inhibitors: Antimicrobial and hemolytic activities against uropathogenic isolates with molecular docking study.
    Ammar YA, Micky JA, Aboul-Magd DS, Abd El-Hafez SMA, Hessein SA, Ali AM, Ragab A.
    Chem Biol Drug Des; 2023 Feb 14; 101(2):245-270. PubMed ID: 36305722
    [Abstract] [Full Text] [Related]

  • 12. Discovery of New Schiff Bases Tethered Pyrazole Moiety: Design, Synthesis, Biological Evaluation, and Molecular Docking Study as Dual Targeting DHFR/DNA Gyrase Inhibitors with Immunomodulatory Activity.
    Hassan AS, Askar AA, Naglah AM, Almehizia AA, Ragab A.
    Molecules; 2020 Jun 02; 25(11):. PubMed ID: 32498469
    [Abstract] [Full Text] [Related]

  • 13. Synthesis, Antimicrobial Activity and Molecular Docking of Novel Thiourea Derivatives Tagged with Thiadiazole, Imidazole and Triazine Moieties as Potential DNA Gyrase and Topoisomerase IV Inhibitors.
    Hashem HE, Amr AEE, Nossier ES, Elsayed EA, Azmy EM.
    Molecules; 2020 Jun 15; 25(12):. PubMed ID: 32549386
    [Abstract] [Full Text] [Related]

  • 14. Design of (quinolin-4-ylthio)carboxylic acids as new Escherichia coli DNA gyrase B inhibitors: machine learning studies, molecular docking, synthesis and biological testing.
    Metelytsia L, Hodyna D, Dobrodub I, Semenyuta I, Zavhorodnii M, Blagodatny V, Kovalishyn V, Brazhko O.
    Comput Biol Chem; 2020 Apr 15; 85():107224. PubMed ID: 32018168
    [Abstract] [Full Text] [Related]

  • 15. Synthesis of novel 2-aminobenzothiazole derivatives as potential antimicrobial agents with dual DNA gyrase/topoisomerase IV inhibition.
    Ismail MMF, Abdulwahab HG, Nossier ES, El Menofy NG, Abdelkhalek BA.
    Bioorg Chem; 2020 Jan 15; 94():103437. PubMed ID: 31812260
    [Abstract] [Full Text] [Related]

  • 16. Design, synthesis and molecular modeling studies of new series of s-triazine derivatives as antimicrobial agents against multi-drug resistant clinical isolates.
    Haiba NS, Khalil HH, Moniem MA, El-Wakil MH, Bekhit AA, Khattab SN.
    Bioorg Chem; 2019 Aug 15; 89():103013. PubMed ID: 31174040
    [Abstract] [Full Text] [Related]

  • 17. Design, synthesis, antimicrobial activity and molecular docking studies of some novel di-substituted sulfonylquinoxaline derivatives.
    Ammar YA, Farag AA, Ali AM, Ragab A, Askar AA, Elsisi DM, Belal A.
    Bioorg Chem; 2020 Nov 15; 104():104164. PubMed ID: 32896807
    [Abstract] [Full Text] [Related]

  • 18. Chrysin based pyrimidine-piperazine hybrids: design, synthesis, in vitro antimicrobial and in silico E. coli topoisomerase II DNA gyrase efficacy.
    Patel KB, Rajani D, Ahmad I, Patel H, Patel HD, Kumari P.
    Mol Divers; 2024 Jun 15; 28(3):1377-1392. PubMed ID: 37318711
    [Abstract] [Full Text] [Related]

  • 19. Potent antibacterial activity of dihydydropyrimidine-1,3,5-triazines via inhibition of DNA gyrase and antifungal activity with favourable metabolic profile.
    Masih A, Shrivastava JK, Bhat HR, Singh UP.
    Chem Biol Drug Des; 2020 Aug 15; 96(2):861-869. PubMed ID: 32333828
    [Abstract] [Full Text] [Related]

  • 20. Design and synthesis of some novel hybrid molecules based on 4-thiazolidinone bearing pyridine-pyrazole scaffolds: molecular docking and molecular dynamics simulations of its major constituent onto DNA gyrase inhibition.
    Desai NC, Jadeja DJ, Jethawa AM, Ahmad I, Patel H, Dave BP.
    Mol Divers; 2024 Apr 15; 28(2):693-709. PubMed ID: 36750538
    [Abstract] [Full Text] [Related]


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