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Journal Abstract Search


219 related items for PubMed ID: 8681408

  • 1. Design and synthesis of 6-chloro-3,4-dihydro-4-methyl-2H-1,4-benzoxazine-8-carboxamide derivatives as potent serotonin-3 (5-HT3) receptor antagonists.
    Kuroita T, Sakamori M, Kawakita T.
    Chem Pharm Bull (Tokyo); 1996 Apr; 44(4):756-64. PubMed ID: 8681408
    [Abstract] [Full Text] [Related]

  • 2. Benzoxazines. II. Synthesis, conformational analysis, and structure--activity relationships of 3,4-dihydro-2H-1,4-benzoxazine-8-carboxamide derivatives as potent and long-acting serotonin-3 (5-HT3) receptor antagonists.
    Kuroita T, Marubayashi N, Sano M, Kanzaki K, Inaba K, Kawakita T.
    Chem Pharm Bull (Tokyo); 1996 Nov; 44(11):2051-60. PubMed ID: 8945770
    [Abstract] [Full Text] [Related]

  • 3. New 5-HT3 (serotonin-3) receptor antagonists. V. Synthesis and structure-activity relationships of pyrrolo[2,1-c][1,4]benzoxazine-6-carboxamides.
    Kato M, Nishino S, Ito K, Yamakuni H, Takasugi H.
    Chem Pharm Bull (Tokyo); 1995 Aug; 43(8):1358-63. PubMed ID: 7553981
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  • 4. Synthesis and pharmacology of 3,4-dihydro-3-oxo-1,4-benzoxazine-8-carboxamide derivatives, a new class of potent serotonin-3 (5-HT3) receptor antagonists.
    Kawakita T, Kuroita T, Yasumoto M, Sano M, Inaba K, Fukuda T, Tahara T.
    Chem Pharm Bull (Tokyo); 1992 Mar; 40(3):624-30. PubMed ID: 1611677
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  • 6. Synthesis of a new class of 2,3-dihydro-2-oxo-1H-benzimidazole-1-carboxylic acid derivatives as highly potent 5-HT3 receptor antagonists.
    Turconi M, Nicola M, Quintero MG, Maiocchi L, Micheletti R, Giraldo E, Donetti A.
    J Med Chem; 1990 Aug; 33(8):2101-8. PubMed ID: 1695682
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  • 9. Development of potent serotonin-3 (5-HT3) receptor antagonists. I. Structure-activity relationships of 2-alkoxy-4-amino-5-chlorobenzamide derivatives.
    Harada H, Morie T, Hirokawa Y, Yoshida N, Kato S.
    Chem Pharm Bull (Tokyo); 1995 Aug; 43(8):1364-78. PubMed ID: 7553982
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  • 10. Antagonistic activity of Y-25130 on 5-HT3 receptors.
    Sato N, Sakamori M, Haga K, Takehara S, Setoguchi M.
    Jpn J Pharmacol; 1992 Aug; 59(4):443-8. PubMed ID: 1331590
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  • 11. Synthesis and structure-activity relationships of 4-amino-5-chloro-N-(1,4-dialkylhexahydro-1,4-diazepin-6-yl)-2-methoxybenzamide derivatives, novel and potent serotonin 5-HT3 and dopamine D2 receptors dual antagonist.
    Hirokawa Y, Harada H, Yoshikawa T, Yoshida N, Kato S.
    Chem Pharm Bull (Tokyo); 2002 Jul; 50(7):941-59. PubMed ID: 12130853
    [Abstract] [Full Text] [Related]

  • 12. New 5-HT3 (serotonin-3) receptor antagonists. IV. Synthesis and structure-activity relationships of azabicycloalkaneacetamide derivatives.
    Kato M, Ito K, Nishino S, Yamakuni H, Takasugi H.
    Chem Pharm Bull (Tokyo); 1995 Aug; 43(8):1351-7. PubMed ID: 7553980
    [Abstract] [Full Text] [Related]

  • 13. The function of 5-HT3 receptors on colonic transit in rats.
    Haga K, Asano K, Fukuda T, Kobayakawa T.
    Obes Res; 1995 Dec; 3 Suppl 5():801S-810S. PubMed ID: 8653566
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  • 14. Comparison of potencies of 5-HT3 receptor antagonists at inhibiting aversive behavior to illumination and the von Bezold-Jarisch reflex in the mouse.
    Eglen RM, Lee CH, Khabbaz M, Fontana DJ, Daniels S, Kilfoil T, Wong EH.
    Neuropharmacology; 1994 Feb; 33(2):227-34. PubMed ID: 8035908
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  • 15. Phenylimidazolidin-2-one derivatives as selective 5-HT3 receptor antagonists and refinement of the pharmacophore model for 5-HT3 receptor binding.
    Heidempergher F, Pillan A, Pinciroli V, Vaghi F, Arrigoni C, Bolis G, Caccia C, Dho L, McArthur R, Varasi M.
    J Med Chem; 1997 Oct 10; 40(21):3369-80. PubMed ID: 9341912
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  • 16. GYKI-46 903, a non-competitive antagonist for 5-HT3 receptors.
    Csillik-Perczel V, Bakonyi A, Yemane T, Vitalis B, Horvath E, Solyom S, Szekely JI, Harsing LG.
    Pharmacol Toxicol; 1996 Jul 10; 79(1):32-9. PubMed ID: 8841094
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  • 17. Comparison of the 5-HT3 receptor antagonist properties of ICS 205-930, GR38032F and zacopride.
    Cohen ML, Bloomquist W, Gidda JS, Lacefield W.
    J Pharmacol Exp Ther; 1989 Jan 10; 248(1):197-201. PubMed ID: 2521513
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  • 18. Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed.
    Leurs R, Tulp MT, Menge WM, Adolfs MJ, Zuiderveld OP, Timmerman H.
    Br J Pharmacol; 1995 Oct 10; 116(4):2315-21. PubMed ID: 8564266
    [Abstract] [Full Text] [Related]

  • 19. The enantiomers of zacopride: an intra-species comparison of their potencies in functional and anxiolytic models.
    Bill DJ, Coleman J, Hallett I, Middlefell VC, Rhodes KF, Fletcher A.
    Br J Pharmacol; 1995 Jul 10; 115(5):775-80. PubMed ID: 8548176
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  • 20. Development of potent serotonin-3 (5-HT3) receptor antagonists. II. Structrue-activity relationships of N-(1-benzyl-4-methylhexahydro-1H-1,4- diazepin-6-yl)carboxamides.
    Harada H, Morie T, Hirokawa Y, Terauchi H, Fujiwara I, Yoshida N, Kato S.
    Chem Pharm Bull (Tokyo); 1995 Nov 10; 43(11):1912-30. PubMed ID: 8575032
    [Abstract] [Full Text] [Related]


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