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148 related items for PubMed ID: 8917649

  • 1. Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist.
    Giardinà D, Crucianelli M, Romanelli R, Leonardi A, Poggesi E, Melchiorre C.
    J Med Chem; 1996 Nov 08; 39(23):4602-7. PubMed ID: 8917649
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  • 2. Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.
    Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D.
    Bioorg Med Chem; 2007 Mar 15; 15(6):2334-45. PubMed ID: 17276073
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  • 3. Synthesis, absolute configuration, and biological profile of the enantiomers of trans-[2-(2,6-dimethoxyphenoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (mephendioxan), a potent competitive alpha 1A-adrenoreceptor antagonist.
    Quaglia W, Pigini M, Tayebati SK, Piergentili A, Giannella M, Leonardi A, Taddei C, Melchiorre C.
    J Med Chem; 1996 May 24; 39(11):2253-8. PubMed ID: 8667368
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  • 5. Search for alpha 1-adrenoceptor subtypes selective antagonists: design, synthesis and biological activity of cystazosin, an alpha 1D-adrenoceptor antagonist.
    Minarini A, Budriesi R, Chiarini A, Leonardi A, Melchiorre C.
    Bioorg Med Chem Lett; 1998 Jun 02; 8(11):1353-8. PubMed ID: 9871765
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  • 7. Searching for cyclazosin analogues as alpha(1B)-adrenoceptor antagonists.
    Giardinà D, Polimanti O, Sagratini G, Angeli P, Gulini U, Marucci G, Melchiorre C, Poggesi E, Leonardi A.
    Farmaco; 2003 Jul 02; 58(7):477-87. PubMed ID: 12818686
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  • 8. Absolute configuration of the alpha (1B)-adrenoceptor antagonist (+)-cyclazosin.
    Giardinà D, Sagratini G, Grelli M, Gulini U, Melchiorre C, Antolini L.
    Farmaco; 2004 Dec 02; 59(12):965-9. PubMed ID: 15598431
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  • 9. 1,3-dioxolane-based ligands as a novel class of alpha1-adrenoceptor antagonists.
    Brasili L, Sorbi C, Franchini S, Manicardi M, Angeli P, Marucci G, Leonardi A, Poggesi E.
    J Med Chem; 2003 Apr 10; 46(8):1504-11. PubMed ID: 12672251
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  • 10. Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes.
    Quaglia W, Pigini M, Piergentili A, Giannella M, Marucci G, Poggesi E, Leonardi A, Melchiorre C.
    J Med Chem; 1999 Jul 29; 42(15):2961-8. PubMed ID: 10425105
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  • 11. (+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues.
    Marucci G, Angeli P, Buccioni M, Gulini U, Melchiorre C, Sagratini G, Testa R, Giardinà D.
    Eur J Pharmacol; 2005 Oct 17; 522(1-3):100-7. PubMed ID: 16213480
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  • 14. 1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: structure-affinity/activity relationship at alpha1-adrenoceptor subtypes and at 5-HT1A receptors.
    Franchini S, Prandi A, Baraldi A, Sorbi C, Tait A, Buccioni M, Marucci G, Cilia A, Pirona L, Fossa P, Cichero E, Brasili L.
    Eur J Med Chem; 2010 Sep 17; 45(9):3740-51. PubMed ID: 20605276
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  • 15. Chiral analogues of (+)-cyclazosin as potent α1B-adrenoceptor selective antagonist.
    Sagratini G, Buccioni M, Marucci G, Poggesi E, Skorski M, Costanzi S, Giardinà D.
    Bioorg Med Chem; 2018 Jul 23; 26(12):3502-3513. PubMed ID: 29784274
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  • 16. Comparison of the binding affinity of some newly synthesized phenylethanolamine and phenoxypropanolamine compounds at recombinant human beta- and alpha1-adrenoceptor subtypes.
    Ahmed M, Hanaoka Y, Kiso T, Kakita T, Ohtsubo Y, Muramatsu I, Nagatomo T.
    J Pharm Pharmacol; 2005 Jan 23; 57(1):75-81. PubMed ID: 15638996
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  • 17. Actions of terazosin and its enantiomers at subtypes of alpha 1- and alpha 2-adrenoceptors in vitro.
    Hancock AA, Buckner SA, Ireland LM, Knepper SM, Kerwin JF.
    J Recept Signal Transduct Res; 1995 Jan 23; 15(7-8):863-85. PubMed ID: 8673721
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  • 19. Comparative alpha-1 adrenoceptor subtype selectivity and functional uroselectivity of alpha-1 adrenoceptor antagonists.
    Martin DJ, Lluel P, Guillot E, Coste A, Jammes D, Angel I.
    J Pharmacol Exp Ther; 1997 Jul 23; 282(1):228-35. PubMed ID: 9223558
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  • 20. Pharmacological properties of the cloned alpha 1A/D-adrenoceptor subtype are consistent with the alpha 1A-adrenoceptor characterized in rat cerebral cortex and vas deferens.
    Kenny BA, Naylor AM, Greengrass PM, Russell MJ, Friend SJ, Read AM, Wyllie MG.
    Br J Pharmacol; 1994 Apr 23; 111(4):1003-8. PubMed ID: 7913370
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