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23. Two neighboring residues of loop A of the alpha1 subunit point towards the benzodiazepine binding site of GABAA receptors. Tan KR, Baur R, Gonthier A, Goeldner M, Sigel E. FEBS Lett; 2007 Oct 02; 581(24):4718-22. PubMed ID: 17854801 [Abstract] [Full Text] [Related]
28. Modifications of gamma-aminobutyric acidA receptor subunit expression in rat neocortex during tolerance to diazepam. Impagnatiello F, Pesold C, Longone P, Caruncho H, Fritschy JM, Costa E, Guidotti A. Mol Pharmacol; 1996 May 02; 49(5):822-31. PubMed ID: 8622632 [Abstract] [Full Text] [Related]
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32. Characterization of U-97775 as a GABAA receptor ligand of dual functionality in cloned rat GABAA receptor subtypes. Im HK, Im WB, Pregenzer JF, Carter DB, Jacobsen EJ, Hamilton BJ. Br J Pharmacol; 1995 May 02; 115(1):19-24. PubMed ID: 7647975 [Abstract] [Full Text] [Related]
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35. Diazepam enhancement of GABA-gated currents in binary and ternary GABAA receptors: relationship to benzodiazepine binding site density. Granja R, Gunnersen D, Wong G, Valeyev A, Skolnick P. J Mol Neurosci; 1997 Dec 02; 9(3):187-95. PubMed ID: 9481620 [Abstract] [Full Text] [Related]
36. Mutagenesis of the rat alpha1 subunit of the gamma-aminobutyric acid(A) receptor reveals the importance of residue 101 in determining the allosteric effects of benzodiazepine site ligands. Dunn SM, Davies M, Muntoni AL, Lambert JJ. Mol Pharmacol; 1999 Oct 02; 56(4):768-74. PubMed ID: 10496960 [Abstract] [Full Text] [Related]
37. Identification of a residue in the gamma-aminobutyric acid type A receptor alpha subunit that differentially affects diazepam-sensitive and -insensitive benzodiazepine site binding. Derry JM, Dunn SM, Davies M. J Neurochem; 2004 Mar 02; 88(6):1431-8. PubMed ID: 15009644 [Abstract] [Full Text] [Related]
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39. A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity. Buhr A, Sigel E. Proc Natl Acad Sci U S A; 1997 Aug 05; 94(16):8824-9. PubMed ID: 9238062 [Abstract] [Full Text] [Related]
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