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Journal Abstract Search
145 related items for PubMed ID: 9871765
1. Search for alpha 1-adrenoceptor subtypes selective antagonists: design, synthesis and biological activity of cystazosin, an alpha 1D-adrenoceptor antagonist. Minarini A, Budriesi R, Chiarini A, Leonardi A, Melchiorre C. Bioorg Med Chem Lett; 1998 Jun 02; 8(11):1353-8. PubMed ID: 9871765 [Abstract] [Full Text] [Related]
2. Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin. Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D. Bioorg Med Chem; 2007 Mar 15; 15(6):2334-45. PubMed ID: 17276073 [Abstract] [Full Text] [Related]
3. Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist. Giardinà D, Crucianelli M, Romanelli R, Leonardi A, Poggesi E, Melchiorre C. J Med Chem; 1996 Nov 08; 39(23):4602-7. PubMed ID: 8917649 [Abstract] [Full Text] [Related]
4. (+)-Cyclazosin, a selective alpha1B-adrenoceptor antagonist: functional evaluation in rat and rabbit tissues. Marucci G, Angeli P, Buccioni M, Gulini U, Melchiorre C, Sagratini G, Testa R, Giardinà D. Eur J Pharmacol; 2005 Oct 17; 522(1-3):100-7. PubMed ID: 16213480 [Abstract] [Full Text] [Related]
7. (+/-)-Domesticine, a novel and selective alpha1D-adrenoceptor antagonist in animal tissues and human alpha 1-adrenoceptors. Indra B, Matsunaga K, Hoshino O, Suzuki M, Ogasawara H, Muramatsu I, Taniguchi T, Ohizumi Y. Eur J Pharmacol; 2002 Jun 07; 445(1-2):21-9. PubMed ID: 12065190 [Abstract] [Full Text] [Related]
8. WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for alpha(1)-adrenoreceptor subtypes and 5-HT(1A) receptors. Bolognesi ML, Budriesi R, Cavalli A, Chiarini A, Gotti R, Leonardi A, Minarini A, Poggesi E, Recanatini M, Rosini M, Tumiatti V, Melchiorre C. J Med Chem; 1999 Oct 07; 42(20):4214-24. PubMed ID: 10514291 [Abstract] [Full Text] [Related]
9. Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes. Quaglia W, Pigini M, Piergentili A, Giannella M, Gentili F, Marucci G, Carrieri A, Carotti A, Poggesi E, Leonardi A, Melchiorre C. J Med Chem; 2002 Apr 11; 45(8):1633-43. PubMed ID: 11931617 [Abstract] [Full Text] [Related]
11. Receptor binding profile of cyclazosin, a new alpha 1B-adrenoceptor antagonist. Giardinà D, Crucianelli M, Melchiorre C, Taddei C, Testa R. Eur J Pharmacol; 1995 Dec 04; 287(1):13-6. PubMed ID: 8666020 [Abstract] [Full Text] [Related]
12. Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes. Quaglia W, Pigini M, Piergentili A, Giannella M, Marucci G, Poggesi E, Leonardi A, Melchiorre C. J Med Chem; 1999 Jul 29; 42(15):2961-8. PubMed ID: 10425105 [Abstract] [Full Text] [Related]
13. Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for alpha1-adrenoreceptor subtypes. Bolognesi ML, Budriesi R, Chiarini A, Poggesi E, Leonardi A, Melchiorre C. J Med Chem; 1998 Nov 19; 41(24):4844-53. PubMed ID: 9822553 [Abstract] [Full Text] [Related]
16. Characterization of some novel alpha 1-adrenoceptor antagonists in human hyperplastic prostate. Chueh SC, Chern JW, Choong CM, Guh JH, Teng CM. Eur J Pharmacol; 2002 Jun 07; 445(1-2):125-31. PubMed ID: 12065203 [Abstract] [Full Text] [Related]
17. Differential antagonism by conotoxin rho-TIA of contractions mediated by distinct alpha1-adrenoceptor subtypes in rat vas deferens, spleen and aorta. Lima V, Mueller A, Kamikihara SY, Raymundi V, Alewood D, Lewis RJ, Chen Z, Minneman KP, Pupo AS. Eur J Pharmacol; 2005 Jan 31; 508(1-3):183-92. PubMed ID: 15680270 [Abstract] [Full Text] [Related]
18. Different subtypes of alpha 1A-adrenoceptor mediating contraction of rat epididymal vas deferens, rat hepatic portal vein and human prostate distinguished by the antagonist RS 17053. Marshall I, Burt RP, Green GM, Hussain MB, Chapple CR. Br J Pharmacol; 1996 Sep 31; 119(2):407-15. PubMed ID: 8886428 [Abstract] [Full Text] [Related]
19. A-315456: a selective alpha(1D)-adrenoceptor antagonist with minimal dopamine D(2) and 5-HT(1A) receptor affinity. Buckner SA, Milicic I, Daza A, Lynch JJ, Kolasa T, Nakane M, Sullivan JP, Brioni JD. Eur J Pharmacol; 2001 Dec 14; 433(1):123-7. PubMed ID: 11755142 [Abstract] [Full Text] [Related]