BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

207 related articles for article (PubMed ID: 23579486)

  • 1. A new strategy for selective targeting of progesterone receptor with passive antagonists.
    Khan JA; Tikad A; Fay M; Hamze A; Fagart J; Chabbert-Buffet N; Meduri G; Amazit L; Brion JD; Alami M; Lombès M; Loosfelt H; Rafestin-Oblin ME
    Mol Endocrinol; 2013 Jun; 27(6):909-24. PubMed ID: 23579486
    [TBL] [Abstract][Full Text] [Related]  

  • 2. The nuclear corepressors NCoR and SMRT are key regulators of both ligand- and 8-bromo-cyclic AMP-dependent transcriptional activity of the human progesterone receptor.
    Wagner BL; Norris JD; Knotts TA; Weigel NL; McDonnell DP
    Mol Cell Biol; 1998 Mar; 18(3):1369-78. PubMed ID: 9488452
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New antiprogestins with partial agonist activity: potential selective progesterone receptor modulators (SPRMs) and probes for receptor- and coregulator-induced changes in progesterone receptor induction properties.
    Giannoukos G; Szapary D; Smith CL; Meeker JE; Simons SS
    Mol Endocrinol; 2001 Feb; 15(2):255-70. PubMed ID: 11158332
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Anti-Tumoral Effects of Anti-Progestins in a Patient-Derived Breast Cancer Xenograft Model.
    Esber N; Cherbonnier C; Resche-Rigon M; Hamze A; Alami M; Fagart J; Loosfelt H; Lombès M; Chabbert-Buffet N
    Horm Cancer; 2016 Apr; 7(2):137-47. PubMed ID: 26941094
    [TBL] [Abstract][Full Text] [Related]  

  • 5. The partial agonist activity of antagonist-occupied steroid receptors is controlled by a novel hinge domain-binding coactivator L7/SPA and the corepressors N-CoR or SMRT.
    Jackson TA; Richer JK; Bain DL; Takimoto GS; Tung L; Horwitz KB
    Mol Endocrinol; 1997 Jun; 11(6):693-705. PubMed ID: 9171233
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Molecular determinants of the recognition of ulipristal acetate by oxo-steroid receptors.
    Petit-Topin I; Fay M; Resche-Rigon M; Ulmann A; Gainer E; Rafestin-Oblin ME; Fagart J
    J Steroid Biochem Mol Biol; 2014 Oct; 144 Pt B():427-35. PubMed ID: 25204619
    [TBL] [Abstract][Full Text] [Related]  

  • 7. A nuclear receptor corepressor modulates transcriptional activity of antagonist-occupied steroid hormone receptor.
    Zhang X; Jeyakumar M; Petukhov S; Bagchi MK
    Mol Endocrinol; 1998 Apr; 12(4):513-24. PubMed ID: 9544987
    [TBL] [Abstract][Full Text] [Related]  

  • 8. A structural and in vitro characterization of asoprisnil: a selective progesterone receptor modulator.
    Madauss KP; Grygielko ET; Deng SJ; Sulpizio AC; Stanley TB; Wu C; Short SA; Thompson SK; Stewart EL; Laping NJ; Williams SP; Bray JD
    Mol Endocrinol; 2007 May; 21(5):1066-81. PubMed ID: 17356170
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Partial agonist activity of the progesterone receptor antagonist RU486 mediated by an amino-terminal domain coactivator and phosphorylation of serine400.
    Wardell SE; Narayanan R; Weigel NL; Edwards DP
    Mol Endocrinol; 2010 Feb; 24(2):335-45. PubMed ID: 20008003
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Progesterone receptor and the mechanism of action of progesterone antagonists.
    Edwards DP; Altmann M; DeMarzo A; Zhang Y; Weigel NL; Beck CA
    J Steroid Biochem Mol Biol; 1995 Jun; 53(1-6):449-58. PubMed ID: 7626494
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Coactivator/corepressor ratios modulate PR-mediated transcription by the selective receptor modulator RU486.
    Liu Z; Auboeuf D; Wong J; Chen JD; Tsai SY; Tsai MJ; O'Malley BW
    Proc Natl Acad Sci U S A; 2002 Jun; 99(12):7940-4. PubMed ID: 12048256
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Discovery of a novel mechanism of steroid receptor antagonism: WAY-255348 modulates progesterone receptor cellular localization and promoter interactions.
    Yudt MR; Russo LA; Berrodin TJ; Jelinsky SA; Ellis D; Cohen JC; Cooch N; Haglund E; Unwalla RJ; Fensome A; Wrobel J; Zhang Z; Nagpal S; Winneker RC
    Biochem Pharmacol; 2011 Dec; 82(11):1709-19. PubMed ID: 21854761
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Agonist and antagonists induce homodimerization and mixed ligand heterodimerization of human progesterone receptors in vivo by a mammalian two-hybrid assay.
    Leonhardt SA; Altmann M; Edwards DP
    Mol Endocrinol; 1998 Dec; 12(12):1914-30. PubMed ID: 9849965
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Ligand-dependent cross-talk between steroid and thyroid hormone receptors. Evidence for common transcriptional coactivator(s).
    Zhang X; Jeyakumar M; Bagchi MK
    J Biol Chem; 1996 Jun; 271(25):14825-33. PubMed ID: 8662980
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Distinct temporal and spatial activities of RU486 on progesterone receptor function in reproductive organs of ovariectomized mice.
    Han SJ; Tsai SY; Tsai MJ; O'Malley BW
    Endocrinology; 2007 May; 148(5):2471-86. PubMed ID: 17303655
    [TBL] [Abstract][Full Text] [Related]  

  • 16. The opposing transcriptional activities of the two isoforms of the human progesterone receptor are due to differential cofactor binding.
    Giangrande PH; Kimbrel EA; Edwards DP; McDonnell DP
    Mol Cell Biol; 2000 May; 20(9):3102-15. PubMed ID: 10757795
    [TBL] [Abstract][Full Text] [Related]  

  • 17. The novel progesterone receptor antagonists RTI 3021-012 and RTI 3021-022 exhibit complex glucocorticoid receptor antagonist activities: implications for the development of dissociated antiprogestins.
    Wagner BL; Pollio G; Giangrande P; Webster JC; Breslin M; Mais DE; Cook CE; Vedeckis WV; Cidlowski JA; McDonnell DP
    Endocrinology; 1999 Mar; 140(3):1449-58. PubMed ID: 10067874
    [TBL] [Abstract][Full Text] [Related]  

  • 18. p38 and p42/44 MAPKs differentially regulate progesterone receptor A and B isoform stabilization.
    Khan JA; Amazit L; Bellance C; Guiochon-Mantel A; Lombès M; Loosfelt H
    Mol Endocrinol; 2011 Oct; 25(10):1710-24. PubMed ID: 21816898
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Agonist and antagonist-induced qualitative and quantitative alterations of progesterone receptor from breast cancer cells.
    Hurd C; Nag K; Khattree N; Alban P; Dinda S; Moudgil VK
    Mol Cell Biochem; 1999 Sep; 199(1-2):49-56. PubMed ID: 10544951
    [TBL] [Abstract][Full Text] [Related]  

  • 20. The X-ray structure of RU486 bound to the progesterone receptor in a destabilized agonistic conformation.
    Raaijmakers HC; Versteegh JE; Uitdehaag JC
    J Biol Chem; 2009 Jul; 284(29):19572-9. PubMed ID: 19372222
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.